| ID | Name | Organism | Chains bound to carbohydrates |
|---|---|---|---|
| 1 | Histone-lysine N-methyltransferase, H3 lysine-79 specific Q8TEK3 (DOT1L_HUMAN) |
Homo sapiens | 1 chain bound to carbohydrates Chain A: 1 binding site |
| ID | Description | N° of binding sites | Bound to chains | Binding affinity |
|---|---|---|---|---|
| 2 | 5'-[{cis-3-[2-(5-tert-butyl-1h-benzimidazol-2-yl)ethyl]cyclobutyl}(propan-2-yl)amino]-5'-deoxyadenosine | 1 (1 molecule) | A | -logKd/Ki=10.10, Ki=0.08nM (PDBbind-CN),Ki=0.080000nM, IC50=<0.100000nM (BindingDB) |